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10-4167

Alpelisib

Size

£139.00

SKU:
10-4167
Additional Names:
BYL719|NVP-BYL719
Physical State:
Solid
Molecular Weight:
441.47
Purity:
>98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
1217486-61-7
Immunogen:
Kinase
Extra Details:
Alpelisib is a potent and selective (IC50s = 7.4 nM PI3KA Alpha; 2.2 uM PI3KB Beta; 1.2 uM PI3KID Delta; 50-fold selectivity against 442 tested kinases) PI3KA Alpha inhibitor.1 Approved for use in the treatment of HR(+), HER2(-), PIK3CA-mutated breast cancer. Alpelisib has been used in combination with various chemotherapeutics to treat ovarian2, colorectal3, kidney4, bladder5, and head and neck6 cancers.
Shipping Conditions:
Ambient