10-3990
PF-05089771
Size
£158.00
- SKU:
- 10-3990
- Additional Names:
- PF771
- Physical State:
- Solid
- Molecular Weight:
- 500.34
- Purity:
- 98%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 1235403-62-9
- Immunogen:
- Ion channel
- Extra Details:
- Potent and selective inhibitor of the voltage gated sodium channel 1.7 (Nav1.7).1,3 It is a state-dependent inhibitor with IC50 = 11 nM for the half-inactivated channels and IC50 ~ 10 uM for resting channels.1 Equipotent for human, monkey, dog, and mouse channels but 15x less potent for rat channels. Interacts equally with fast and slow inactivated Nav1.7 channels.2
- Shipping Conditions:
- Ambient