Skip to content

Download Spec Sheet

download
  1. Shop all
  2. Antagonists

10-2957

Cinacalcet HCl

Size

£149.00

SKU:
10-2957
Additional Names:
AMG 073|KRN 1493|Mimpara|Sensipar
Physical State:
Solid
Molecular Weight:
393.88
Purity:
>98%
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
364782-34-3
Immunogen:
GPCR
Extra Details:
Cinacalcet (364782-34-3) is a calcimimetic that allosterically activates the calcium-sensing receptor (CaSR; EC50 = 79.4 nM in HEK 293T cells expressing CaSR).1-3 It lowers plasma parathyroid hormone in hemodialysis patients with secondary hyperparathyroidism.4 Cinacalcet has been used to treat parathyroid carcinoma.5
Shipping Conditions:
Ambient