10-2177
Tofacitinib

Size
£158.00
- SKU:
- 10-2177
- Additional Names:
- CP-690550|Tasocitinib
- Physical State:
- Solid
- Molecular Weight:
- 312.37
- Purity:
- 99%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 477600-75-2
- Immunogen:
- Kinase
- Extra Details:
- Potent pan-JAK inhibitor, IC50s=1, 20 and 112 nM for JAK3, JAK2 and JAK1 respectively.1 Displays potent antiinflammatory2 and immunosuppressant3 activity. Promotes a white-to-brown metabolic metabolic conversion in human adipoctes.4 In therapeutic use for rheumatoid arthritis.5
- Shipping Conditions:
- Ambient
