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10-2177

Tofacitinib

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£158.00

SKU:
10-2177
Additional Names:
CP-690550|Tasocitinib
Physical State:
Solid
Molecular Weight:
312.37
Purity:
99%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
477600-75-2
Immunogen:
Kinase
Extra Details:
Potent pan-JAK inhibitor, IC50s=1, 20 and 112 nM for JAK3, JAK2 and JAK1 respectively.1 Displays potent antiinflammatory2 and immunosuppressant3 activity. Promotes a white-to-brown metabolic metabolic conversion in human adipoctes.4 In therapeutic use for rheumatoid arthritis.5
Shipping Conditions:
Ambient