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10-2125

CI-994

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£137.00

SKU:
10-2125
Additional Names:
GOE-5549|N-acetyl-dinaline|PD-123654|Tacedinaline
Physical State:
Solid
Molecular Weight:
269.30
Purity:
98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
112522-64-2
Immunogen:
Protein deacetylase
Extra Details:
Orally active histone deacetylase (HDAC) inhibitor, IC50 = 0.9, 0.9, 1.2 and >20 uM for HDAC1, HDAC2, HDAC3 and HDAC8 respectively.1 Mediates G1 cell cycle arrest, inhibits proliferation and induces apoptosis in vitro and in vivo.2,3 Increases neuroplasticity during memory extinction.4 Protects beta cells from cytokine-induced apoptosis.4
Shipping Conditions:
Ambient