10-2125
CI-994

Size
£137.00
- SKU:
- 10-2125
- Additional Names:
- GOE-5549|N-acetyl-dinaline|PD-123654|Tacedinaline
- Physical State:
- Solid
- Molecular Weight:
- 269.30
- Purity:
- 98%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 112522-64-2
- Immunogen:
- Protein deacetylase
- Extra Details:
- Orally active histone deacetylase (HDAC) inhibitor, IC50 = 0.9, 0.9, 1.2 and >20 uM for HDAC1, HDAC2, HDAC3 and HDAC8 respectively.1 Mediates G1 cell cycle arrest, inhibits proliferation and induces apoptosis in vitro and in vivo.2,3 Increases neuroplasticity during memory extinction.4 Protects beta cells from cytokine-induced apoptosis.4
- Shipping Conditions:
- Ambient
