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10-1351

WP-1130

Size

£153.00

SKU:
10-1351
Additional Names:
Degrasyn
Physical State:
Solid
Molecular Weight:
384.28
Purity:
98%
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
856243-80-6
Immunogen:
DUB (Deubiquitinating enzyme)
Extra Details:
A novel DUB inhibitor directly inhibiting USP9x, USP5, USP14 and UCH37 inducing rapid accumulation of polyubiquitinated proteins. Triggers tumor cell apoptosis.1 Blocks Jak2 signaling via Jak2 ubiquitination.2 Causes ablation of the oncogenic transcription factor ERG in prostate cancer cells.3
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Ambient