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10-1126

Vinpocetine

Size

£149.00

SKU:
10-1126
Physical State:
Solid
Molecular Weight:
350.45
Purity:
98%
Storage Conditions:
RT
Supplier:
Focus Biomolecules
CAS Number:
42971-09-5
Immunogen:
PDE (Phosphodiesterase)
Extra Details:
Phosphodiesterase PDE1 inhibitor (IC50=21 uM)1. Also blocks voltage-gated Na+ channels, IC50=44.2 uM (potency similar to phenytoin), a mechanism which may contribute to its neuroprotective and anticonvulsant activity2. It reduces inflammatory IL-1B Beta and TNF-A Alpha expression in rat hippocampus3. Displays beneficial effects in a rat model of cerebral ischemia-reperfusion injury4. Exerts neuroprotective effects by suppressing microglial inflammation5.
Shipping Conditions:
Ambient