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Product Sizes
5 mg
£158.00
10-1539-5MG
25 mg
£281.00
10-1539-25MG
About this Product
SKU:
10-1539
Additional Names:
trans-ISRIB
CAS Number:
1597403-47-8
Extra Details:
Integrated stress response inhibitor. Potently reverses the effects of initiation factor 2A Alpha (eIF2A Alpha) phosphorylation, IC50=5 nM.1 Enhances spatial and fear-associated learning in mice and enhances cognitive function.1,2 Mechanism of action involves activation of eiF2B Beta.3 Suppresses ER stress-induced inflammatory gene expression.4 Potently attenuates amyloid B Beta-induced neuronal cell death (12.5-25 nM) with no effect on amyloid B Beta production.5 Reverses hippocampal-dependent cognitive deficits induced by traumatic brain injury in two different injury mouse models.6
Immunogen:
ER/Golgi|Ribosome|UPR (Unfolded protein response)
Molecular Weight:
451.34
Physical State:
Solid
Purity:
98%
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors
Sell Sheet 1:
View Sell Sheet Here