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E3317-75

Enzastaurin, Free Base

Größe

£209.00

SKU:
E3317-75
Molekulargewicht:
515.6
Reinheit:
~99%
Lagerbedingungen:
-20°C
Hersteller:
United States Biological
CAS Number:
170364-57-5
Format:
Supplied as a red-orange powder.
Weitere Details:
Enzastaurin inhibits PKCb, PKCa, PKCy and PKCe with IC50's of 0.006, 0.039, 0.083 and 0.110uM, respectively. Enzastaurin apparently inhibits tumor growth via multiple mechanisms: suppression of tumor cell proliferation, induction of tumor cell apoptosis and inhibition of tumor-induced angiogenesis. Solubility: Soluble in DMSO at 7.1mg/ml with warming; very poorly soluble in ethanol; very poorly soluble in water; maximum solubility in plain water is estimated to be about 1-10uM; buffers, serum, or other additives may increase or decrease the aqueous solubility. Storage and Stability: May be stored at RT for short-term only. Long-term storage is recommended at -20°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
Versandbedingungen:
Blue Ice