DY 268

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£442.00

SKU:: 447755
Molekulargewicht:: 560.66
Reinheit:: ≥98% (HPLC)
Lagerbedingungen:: 4°C
Hersteller:: United States Biological
CAS Number:: 1609564-75-1
Format:: White to off-white powder
Weitere Details:: DY-268 is a trisubstituted-pyrazol carboamide based compound that acts as a potent FXR antagonist (IC50 = 7.5 nM). It does not display any FXR agonistic activity and cytotoxicity. Synonyms: 1-(3-Methoxybenzyl)-N-(4-methyl-3-(morpholinosulfonyl)phenyl)-3-(p-tolyl)-1H-pyrazole-4-carboxamide; 1-[(3-Methoxyphenyl)methyl]-N-[4-methyl-3-(4-morpholinylsulfonyl)phenyl]-3-(4-methylphenyl)-1H-pyrazole-4-carboxamide CAS No: 1609564-75-1 Molecular Formula: C₃₀H₃₂N₄O₅S Molecular Weight: 560.66 Solubility: DMSO, 50-100mg/ml Biological Activity: Potent FXR antagonist (IC50 = 7.5 nM). Exhibits no detectable cytotoxicity in cell-based assays. Appearance: White to off-white powder Purity ≥98% (HPLC) Storage and Stability: Store at 4°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.