SB-705498

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£163.00

SKU:: 10-3985
Physischer Zustand:: Solid
Molekulargewicht:: 429.24
Reinheit:: 98%
Aufreinigung:: HPLC Purified
Lagerbedingungen:: -20[o]C
Hersteller:: Focus Biomolecules
CAS Number:: 501951-42-4
Immunogen:: Ion channel
Weitere Details:: Potent and selective antagonist of the TRPV1 receptor (IC50's for receptor induction method: Capsaicin = 3 nM; Acid (pH5.3) = pIC50 7.1, and Heat = 6 nM) with activity in human, rat, and guinea pig receptors.1,2 SB-705498s activity is voltage dependent and shows >100 fold selectivity over the closely related TRPM8 receptor.2