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10-1531

DC260126

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£147.00

SKU:
10-1531
Physischer Zustand:
Solid
Molekulargewicht:
307.37
Reinheit:
98%
Aufreinigung:
HPLC Purified
Lagerbedingungen:
-20[o]C
Hersteller:
Focus Biomolecules
CAS Number:
346692-04-4
Immunogen:
GPCR
Weitere Details:
A GPR40 receptor antagonist1. Suppresses fatty acid-induced elevation of intracellular Ca++. Inhibits palmitic acid potentiated glucose-stimulated insulin secretion in Min6 pancreatic B Beta cells in vitro. Lowers serum insulin levels, increases insulin sensitivity2 in obese Zucker rats (6 mg/kg)2. Reduces pancreatic B Beta cell apoptosis in obese diabetic (db/db) rats3. Protects Min6 B Beta cells from palmitic acid-induced ER stress and apoptosis4
Versandbedingungen:
Ambient