10-1198
GSK-1016790A
Größe
£166.00
- SKU:
- 10-1198
- Physischer Zustand:
- Solid
- Molekulargewicht:
- 655.62
- Reinheit:
- 98%
- Lagerbedingungen:
- -20[o]C
- Hersteller:
- Focus Biomolecules
- CAS Number:
- 942206-85-1
- Immunogen:
- Ion channel
- Weitere Details:
- A novel and potent TRPV4 channel agonist. GSK1016790A induced Ca2+ influx in mouse and human TRPV4 expressing HEK cells (EC50 values of 18 and 2.1 nM, respectively), and evoked a dose-dependent activation of TRPV4 whole-cell currents at concentrations above 1 nM. It is 300-fold more potent than 4A Alpha-PDD and is a valuable tool for investigating the role of TRPV4 in physiological processes.
- Versandbedingungen:
- Ambient