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5 mg
£206,00
10-5507-5MG
25 mg
£474,00
10-5507-25MG
Über dieses Produkt
SKU:
10-5507
CAS Number:
294646-77-8
Weitere Details:
Second generation analog of roscovitine which inhibits cyclin-dependent kinases with increased potency, Cdk1/cyclin B, Cdk2/cyclin A, Cdk2/cyclin E, Cdk5, p25, and Cdk9/cyclin T, IC50s=0.09, 0.072, 0.041, 0.11 and 0.18 M respectively.1,2 Acts as a molecular glue degrader that depletes cyclin K.3 CR8 displays neuroprotective effects in various models including traumatic brain injury.4
Immunogen:
Kinase|Molecular glue
Molekulargewicht:
540.91
Physischer Zustand:
Solid
Reinheit:
98%
Aufreinigung:
HPLC Purified
Versandbedingungen:
Ambient
Lagerbedingungen:
-20[o]C
Hersteller:
Focus Biomolecules
Typ:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors
Sell Sheet 1:
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