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5 mg
£138,00
10-4388-5MG
25 mg
£195,00
10-4388-25MG
Über dieses Produkt
SKU:
10-4388
CAS Number:
228559-41-9
Weitere Details:
Very potent (IC50 = 0.9 nM) inhibitor of vascular endothelial growth factor receptor 2 (VEGFR-2).1 It also inhibited PDGFRA Alpha (IC50 = 67 nM), c-Kit (IC50 = 40 nM), and FGFR2 (IC50 = 170 nM). Ki8751 completely suppressed HUVEC growth at 1 nM. Ki8751 completely inhibited tumor growth in LC-6 human tumor xenografts @ 5mg/kg. Ki8751 displayed anti-influenza A and B activity via disruption of virus entry in a PDGFRB Beta/GM3-dependent manner.2
Immunogen:
Kinase
Molekulargewicht:
469.42
Physischer Zustand:
Solid
Reinheit:
>98%
Aufreinigung:
HPLC Purified
Versandbedingungen:
Ambient
Lagerbedingungen:
-20[o]C
Hersteller:
Focus Biomolecules
Typ:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors