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5 mg
£168,00
10-4018-5MG
25 mg
£310,00
10-4018-25MG
Über dieses Produkt
SKU:
10-4018
CAS Number:
1982372-88-2
Weitere Details:
A-196 (1982372-88-2) is a potent and selective (over 29 other methyltransferases) inhibitor of the protein lysine methyltransferases SUV420H1(IC50 = 25 nM) and SUV420H2 (IC50 = 144 nM). It substantially inhibited non-homologous end-joining (NHEJ)-directed DNA repair but not homology-directed repair(HDR) in cells treated with ionizing radiation. A-196 is active in cells and displayed no toxicity in several cell lines.
Immunogen:
Protein methyltransferase
Molekulargewicht:
359.25
Physischer Zustand:
Solid
Reinheit:
98%
Versandbedingungen:
Ambient
Lagerbedingungen:
-20[o]C
Hersteller:
Focus Biomolecules
Typ:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors
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Sell Sheet 2:
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