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Produktgrößen
1 mg
£177,00
10-3958-1MG
5 mg
£334,00
10-3958-5MG
Über dieses Produkt
SKU:
10-3958
CAS Number:
2102501-84-6
Weitere Details:
PF-06835919 is a potent (IC50 = 10 nM KHK-C; 170 nM KHK-A) inhibitor of ketohexokinase (KHK), the first enzyme in the fructose metabolic cascade.1 It displayed high selectivity against other sugar kinases. PF-06835919 prevented hyperinsulinemia, hypertriglyceridemia, and hepatic steatosis in fructose-fed rats.2 The increased tumor proliferation effect of fructose in CaSki cells was inhibited by PF-06835919.3 An interesting new tool to study metabolic and fatty liver diseases.
Immunogen:
Cytochrome/MDR|Sugar kinase
Molekulargewicht:
356.35
Physischer Zustand:
Solid
Reinheit:
>98%
Aufreinigung:
HPLC Purified
Versandbedingungen:
Ambient
Lagerbedingungen:
-20[o]C
Hersteller:
Focus Biomolecules
Typ:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors